C.A. Anderson

University of Oxford

Papers

3

Total Citations

16

H-Index

3

About

C.A. Anderson is a pioneering structural biologist and medicinal chemist whose work is revolutionizing fragment-based drug discovery. Their research centers on overcoming the critical bottleneck in this field: efficiently progressing weakly binding fragment hits into potent lead compounds. Anderson’s major contribution is the development of **Binding-Site Purification of Actives (B-SPA)**, a groundbreaking methodology that integrates multi-step array synthesis with high-throughput crystallography. This approach, detailed in their most-cited 2025 paper (9 citations), enables the rapid, large-scale exploration of chemical space directly within the protein binding site, bypassing traditional, time-consuming purification steps. Complementing this, their 2023 work demonstrated a low-cost, robotics-driven workflow for high-throughput crystallography, making structural data collection on crude reaction mixtures both accessible and efficient. With combined citations exceeding 15, Anderson’s innovations are directly addressing a long-standing “dormant” potential in fragment approaches, offering a credible and scalable path to drug leads. Their work stands as a transformative achievement, promising to accelerate the discovery of new therapeutics by turning fragment screening into a truly high-throughput progression engine.

Research Focus

Key Achievements

3
H-Index
3
Papers
16
Total Citations
5
Avg Citations/Paper
🏆 Most Cited Paper
Binding‐Site Purification of Actives (B‐SPA) Enables Efficient Large‐Scale Progression of Fragment Hits by Combining Multi‐Step Array Synthesis With HT Crystallography
9 citations · 2025
📈 Most Prolific Year: 2025 (1 Papers)
🤝 Key Collaborators: 17
🏛 Institutions: University of Oxford

Top Papers

  1. 1
  2. 2
  3. 3

Key Collaborators

Contact & Links

Available for collaboration
Content generated · 13 days ago