Agonist

A Proteomic Microarray Approach for Exploring Ligand-initiated Nuclear Hormone Receptor Pharmacology, Receptor Selectivity, and Heterodimer Functionality

Sung Hoon Kim, Anobel Tamrazi, Kathryn E. Carlson, John A. Katzenellenbogen

Citations: 41 • 2004

Identification of metabotropic glutamate receptor antagonists using an automated high-throughput screening system

Peter Hodder, Jason Cassaday, Richard Peltier, Kurtis Berry, James Inglese, Bradley P. Feuston, Chris Culberson, Leo Bleicher, Nicholas D. P. Cosford, Chris Bayly, Carla M. Suto, Mark A. Varney, Berta Strulovici

Citations: 39 • 2003

Molecular and Physiological Evidence for Functional γ-Aminobutyric Acid (GABA)-C Receptors in Growth Hormone-secreting Cells

Katia Gamel-Didelon, Lars Kunz, Karl J. Föhr, Manfred Gratzl, Artur Mayerhofer

Citations: 34 • 2003

Application of Division Arrest Technology to Cell-Based HTS: Comparison with Frozen and Fresh Cells

Priya Kunapuli, Wei Zheng, Michael J. Weber, Kelli Solly, Rebecca Mull, Michael Platchek, Mei Cong, Zhong Zhong, Berta Strulovici

Citations: 33 • 2005

Novel equilibrium-point control of agonist-antagonist system with pneumatic artificial muscles

Yohei Ariga, Hang Pham, Mitsunori Uemura, Hiroaki Hirai, Fumio Miyazaki

Citations: 32 • 2012

Prostaglandin-Stimulated Adenylyl Cyclase Activity Via a Pharmacologically Defined EP ₂ Receptor in Human Nonpigmented Ciliary Epithelial Cells

Julie Y. Crider, Brenda Walker Griffin, Naj Sharif

Citations: 26 • 1998

Simplified procedures for the determination of fenoldopam and its metabolites in human plasma by high-performance liquid chromatography with electrochemical detection: comparison of manual and robotic sample preparation methods

Venkata K. Boppana, Kathleen M. Dolce, Matthew J. Cyronak, John A. Ziemniak

Citations: 26 • 1989

A Robotic MCF-7:WS8 Cell Proliferation Assay to Detect Agonist and Antagonist Estrogenic Activity

Chun Yang, Warren Casey, Matthew Stoner, G. J. Kollessery, A. W. Wong, George D. Bittner

Citations: 21 • 2013

Synthesis and biological investigations of [18F]MR18445, a 5-HT3 receptor partial agonist

Tatiana Katounina, Laurent Besret, Martine Dhilly, Marie-Christine Petit-Taboué, Alexandra Barbelivien, Jean‐Claude Baron, François Dauphin, Louisa Barré

Citations: 19 • 1998

NOVEL METHOD FOR THE STUDY OF RECEPTOR Ca²⁺SIGNALLING EXEMPLIFIED BY THE NK1 RECEPTOR

Anders Heding, Christian Elling, Thue W. Schwartz

Citations: 16 • 2002

Virtual agonist-antagonist mechanisms produce biological muscle-like functions

Xiaofeng Xiong, Florentin Wörgötter, Poramate Manoonpong

Citations: 15 • 2014

Recurrence after robotic myomectomy: is it associated with use of GnRH agonist?

Roopina Sangha, Vivek Katukuri, M.M. Palmer, Raminder Khangura

Citations: 10 • 2016

Novel equilibrium-point control of agonist-antagonist system with pneumatic artificial muscles: II. Application to EMG-based human-machine interface for an elbow-joint system

Yohei Ariga, Daisuke Maeda, Hang Pham, Mitsunori Uemura, Hiroaki Hirai, Fumio Miyazaki

Citations: 9 • 2012

Improving Spasticity by Using Botulin Toxin: An Overview Focusing on Combined Approaches

Loredana Raciti, Gianfranco Raciti, Antonio Ammendolia, Alessandro de Sire, Maria Pia Onesta, Rocco Salvatore Calabrò

Citations: 8 • 2024

pnrVSA: human-like actuator with non-linear springs in agonist-antagonist configuration

Luca Fiorio, Alberto Parmiggiani, Bastien Berret, Giulio Sandini, Francesco Nori

Citations: 8 • 2012

High-throughput screening with a miniaturized radioligand competition assay identifies new modulators of human α2-adrenoceptors

Adyary Fallarero, Katariina Pohjanoksa, Gloria Wissel, Ulla-Mari Parkkisenniemi-Kinnunen, Henri Xhaard, Mika Scheinin, Pia Vuorela

Citations: 8 • 2012

Radioligand Binding Assays in the Drug Discovery Process: Potential Pitfalls of High Throughput Screenings

François Noël, Dayde Lane Mendonça da Silva, Luis Eduardo M. Quintas

Citations: 8 • 2011

Development of a Sensitive and HTS-Compatible Reporter Gene Assay for Functional Analysis of Human Adenosine A2a Receptors in CHO-K1 Cells

Yuting Tang, Jing-Qing Luo, Charles R. Fleming, Yan Kong, Gilbert C. Olini, Mary Jo Wildey, Druie Cavender, Keith T. Demarest

Citations: 8 • 2004

A robotic BG1Luc reporter assay to detect estrogen receptor agonists

Matthew Stoner, Chun Yang, George D. Bittner

Citations: 7 • 2014

A Robust and High-Capacity [ ³⁵ S]GTP <i>γ</i> S Binding Assay for Determining Antagonist and Inverse Agonist Pharmacological Parameters of Histamine H ₃ Receptor Ligands

Thomas R. Miller, John L. Baranowski, Brian R. Estvander, David G. Witte, Tracy L. Carr, Arlene M. Manelli, Kathleen M. Krueger, Marlon Cowart, Jorge D. Brioni, Timothy A. Esbenshade

Citations: 7 • 2008