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Novel Multiplexed High Throughput Screening of Selective Inhibitors for Drug-Metabolizing Enzymes Using Human Hepatocytes

Jianhua Liu, Daria I. Vernikovskaya, Gary Bora, Anthony Carlo, Woodrow Burchett, Samantha Jordan, Lloyd Wei Tat Tang, Joy C. Yang, Ye Che, George Chang, Matthew D. Troutman, Li Di

发表年份
2024
引用次数
7

关键词

High-throughput screeningEnzymeCytochrome P450Aldehyde oxidaseDrugDrug discoveryErlotinibComputational biologyVirtual screeningEnzyme inhibition

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